COUP-TFII
Lua error in Module:Infobox_gene at line 53: attempt to index field 'wikibase' (a nil value). COUP-TFII (COUP transcription factor 2), also known as NR2F2 (nuclear receptor subfamily 2, group F, member 2) is a protein that in humans is encoded by the NR2F2 gene.[1][2] The COUP acronym stands for chicken ovalbumin upstream promoter.
Function
[edit | edit source]COUP-TFII plays a critical role in controlling the development of a number of tissues and organs including heart, blood vessels, muscles and limbs.[3][4]
The glucocorticoid receptor (GR) stimulates COUP-TFII-induced transactivation while COUP-TFII represses the GR transcriptional activity.[5][6] COUP-TFII interacts with GATA2 to inhibit adipocyte differentiation.[7]
Structure and ligands
[edit | edit source]The structure of COUP-TF2 LBD is known. Retinoic acid, although not at physiological concentrations, activate this receptor.[8]
Interactions
[edit | edit source]COUP-TFII has been shown to interact with:
References
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External links
[edit | edit source]- Human NR2F1 genome location and NR2F1 gene details page in the UCSC Genome Browser.
- Human NR2F2 genome location and NR2F2 gene details page in the UCSC Genome Browser.
- Overview of all the structural information available in the PDB for UniProt: P24468 (COUP transcription factor 2) at the PDBe-KB.
Further reading
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