PX-3
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| Legal status |
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| Identifiers | |
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| CAS Number | |
| PubChem CID | |
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| E number | {{#property:P628}} |
| CompTox Dashboard (EPA) |
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| ECHA InfoCard | {{#property:P2566}}Lua error in Module:EditAtWikidata at line 29: attempt to index field 'wikibase' (a nil value). |
| Chemical and physical data | |
| Formula | C24H28N4O2 |
| Molar mass | 404.514 g·mol−1 |
| 3D model (JSmol) | |
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PX-3 (also known as APP-CHMINACA) is an indazole-based synthetic cannabinoid. It is a potent agonist of the CB1 receptor with a binding affinity of Ki = 47.6 nM and was originally developed by Pfizer in 2009 as an analgesic medication.[1][2][3][4]
The acronym 'APP' signifies the 'amino', 'phenyl' and 'propanone' elements of the structure. Three related compounds, PX-1 (5F-APP-PICA, SRF-30), PX-2 (5F-APP-PINACA, FU-PX) and APP-FUBINACA were reported by the EMCDDA in late 2014.[5][6]
Legality
[edit | edit source]Sweden's public health agency suggested to classify APP-CHMINACA as hazardous substance on June 1, 2015.[7]
See also
[edit | edit source]References
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- ^ WO 2009106980, "Indazole derivatives"
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