Atagabalin

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Atagabalin
File:Atagabalin.svg
Clinical data
Other namesPD-0200390; PD-200390; PD0200390; PD200390
Routes of
administration
Oral[1]
ATC code
  • none
Identifiers
  • [(3S,4S)-1-(aminomethyl)-3,4-dimethylcyclopentyl]acetic acid
CAS Number
PubChem CID
ChemSpider
UNII
ChEMBL
E number{{#property:P628}}
CompTox Dashboard (EPA)
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Chemical and physical data
FormulaC10H19NO2
Molar mass185.267 g·mol−1
3D model (JSmol)
  • C[C@H]1CC(C[C@@H]1C)(CC(=O)O)CN
  • InChI=1S/C10H19NO2/c1-7-3-10(6-11,4-8(7)2)5-9(12)13/h7-8H,3-6,11H2,1-2H3,(H,12,13)/t7-,8-/m0/s1 checkY
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Atagabalin (INNTooltip International Nonproprietary Name, USANTooltip United States Adopted Name; developmental code name PD-0200390) is a drug developed by Pfizer and related to gabapentin, which similarly binds to the α2δ calcium channels (1 and 2).[1][2] It was under development as a treatment for insomnia, but was discontinued following unsatisfactory trial results.[1][3][4][5][6] The drug reached phase 2 clinical trials for this indication prior to the discontinuation of its development.[1]

See also

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References

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