3-Chloropyridine

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3-Chloropyridine
File:3-chloropyridine.svg
File:3-chloropyridine-from-xtal-3D-bs-17.png
File:3-chloropyridine-from-xtal-3D-sf.png
Names
Preferred IUPAC name
3-Chloropyridine
Identifiers
3D model (JSmol)
ChemSpider
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EC Number
  • 210-955-7
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UNII
  • {{#property:P3117}}Lua error in Module:EditAtWikidata at line 29: attempt to index field 'wikibase' (a nil value).
  • InChI=1S/C5H4ClN/c6-5-2-1-3-7-4-5/h1-4H
    Key: PWRBCZZQRRPXAB-UHFFFAOYSA-N
  • C1=CC(=CN=C1)Cl
Properties
C5H4ClN
Molar mass 113.54 g·mol−1
Appearance colorless liquid
Density 1.194 g/cm3
Boiling point 148 °C (298 °F; 421 K)
1.533
Hazards
GHS labelling:
GHS02: FlammableGHS07: Exclamation mark
Warning
H226, H302, H312, H315, H332
P210, P233, P240, P241, P242, P243, P261, P264, P270, P271, P280, P301+P312, P302+P352, P303+P361+P353, P304+P312, P304+P340, P312, P321, P322, P330, P332+P313, P362, P363, P370+P378, P403+P235, P501
Flash point 65 °C (149 °F; 338 K)
Related compounds
Related compounds
2-Chloropyridine
3-Bromopyridine
Except where otherwise noted, data are given for materials in their standard state (at 25 °C [77 °F], 100 kPa).

3-Chloropyridine is an aryl chloride and isomer of chloropyridine with the formula C5H4ClN. It is a colorless liquid that is mainly used as a building block in organic synthesis.[1]

The compound is a substrate for many coupling processes including the Heck reaction,[2] Suzuki reaction,[3] and Ullmann reaction.[4]

Preparation

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3-Chloropyridine may be prepared by the direct chlorination of pyridine with aluminium chloride used as the catalyst. The yield is 33%.[5]

A less expensive way of preparing 3-chloropyridine consists of the gas phase pyrolysis of a mixture of pyrrole and chloroform in an empty glass tube. The molar ratio of the reagents is one to five. The yields range from 25 to 33%. A little 2-chloropyridine is formed as a side product.[6] The process is thought to be an example of the Ciamician–Dennstedt rearrangement.

Pyrolytic Ciamician-Dennstedt rearrangement leading to 3-chloropyridine
Pyrolytic Ciamician-Dennstedt rearrangement leading to 3-chloropyridine

References

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