Taurolidine/heparin

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Taurolidine/heparin
Combination of
TaurolidineThiadiazinane antimicrobial
HeparinAnti-coagulant
Clinical data
Trade namesDefencath
AHFS/Drugs.comDefencath
License data
Routes of
administration
Intraluminal
ATC code
  • None
Legal status
Legal status
Identifiers
KEGG
E number{{#property:P628}}
CompTox Dashboard (EPA)
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Taurolidine/heparin, sold under the brand name Defencath, is a fixed-dose combination catheter lock solution used for central venous catheter instillation.[1][2] It contains taurolidine, a thiadiazinane antimicrobial; and heparin, an anti-coagulant. Its use is limited to people with kidney failure receiving chronic hemodialysis through a central venous catheter.[1][2]

The most frequently reported adverse reactions include hemodialysis catheter malfunction, hemorrhage/bleeding, nausea, vomiting, dizziness, musculoskeletal chest pain, and thrombocytopenia.[2]

Taurolidine/heparin was approved for medical use in the United States in November 2023.[2][3] The US Food and Drug Administration (FDA) considers it to be a first-in-class medication.[4]

Medical uses

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Taurolidine/heparin is indicated to reduce catheter-related bloodstream infections in adults with kidney failure who are receiving chronic hemodialysis through a central venous catheter.[1][2][5] It is indicated in this limited and specific patient population.[1][2]

History

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Taurolidine/heparin was studied in a single, randomized, active-controlled phase III clinical trial.[2] In this trial, taurolidine/heparin delayed the time it took to acquire a catheter related bloodstream infection.[2] Taurolidine/heparin demonstrated a 71% risk reduction in catheter related bloodstream infections versus the heparin comparator arm (95% confidence interval for risk reduction: 38% to 86%; p value = 0.0006).[2]

References

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  2. ^ a b c d e f g h i Lua error in Module:Citation/CS1/Configuration at line 2172: attempt to index field '?' (a nil value). Public Domain This article incorporates text from this source, which is in the public domain.
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